SPH3127

目录号：SY-112844

SPH3127 (DRI 18) 是一种强有效的、口服具有活力的、新型的 direct renin 抑制剂，其对 recombinant human-renin，human plasma renin activity 的 IC50 值分别为0.4 nM 和 0.45 nM。SPH3127具有抗高血压效果，能够用于研究高血压。

¥2990.00

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(Sar1)-Angiotensin II

目录号：SY-112845

The substitution with Sar at position 1 of angiotensin II resulted in a partial agonistic activity.

¥1035.00

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TD-0212 TFA

目录号：SY-112846

TD-0212 TFA is an orally active dual pharmacology antagonist of angiotensin II type 1 receptor (AT1) and inhibitor of neprilysin (NEP)(pKi of 8.9 for AT1 and a pIC50 of 9.2 for NEP).

¥1552.00

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[Val4] Angiotensin III

目录号：SY-112847

[Val4] Angiotensin III为血管紧张素III类肽，作为Gαq和βarr2反应的高效全激动剂，其pEC50值分别为8.31和8.44。

¥575.00

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TRV-120027

目录号：SY-112848

TRV120027 is a β-arrestin-1-biased agonist of the angiotensin II receptor type 1. TRV120027 inhibits angiotensin II-mediated vasoconstriction and increases cardiomyocyte contractility.

¥641.00

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Pivalopril

目录号：SY-112850

Pivalopril is a new orally active inhibitor of angiotensin-converting enzyme.

¥2346.00

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Olmesartan methyl ester

目录号：SY-112851

Olmesartan methyl ester is an intermediate in the synthesis of Olmesartan medoxomil. Olmesartan medoxomil is a potent and selective angiotensin AT1 receptor antagonist.

¥4600.00

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[Tyr(P)4] Angiotensin II

目录号：SY-112852

[Tyr(P)4] Angiotensin II is a peptide that exerts a multitude of effects on vascular smooth muscle. These effects include the contraction of normal arteries, as well as the induction of hypertrophy or hyperplasia in cultured cells or diseased vessels.

询价

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Valsartan Ethyl Ester

目录号：SY-112853

Valsartan Ethyl Ester is an impurity of Valsartan, an angiotensin II receptor antagonist used for the treatment of high blood pressure and heart failure.

¥702.00

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