PARP1-IN-5

目录号：SY-111067

PARP1-IN-5 是一种低毒、具有口服活性、有效的和有选择性的 PARP-1 抑制剂 (IC50 =14.7 nM)。PARP1-IN-5 可用于癌症研究。

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TNKS-IN-2

目录号：SY-111068

TNKS-IN-2 (compound 40) 是一种有效的选择性 tankyrase (TANKS) 抑制剂，对 TNKS 和 Wnt 的 pIC50 值分别为 8.1、7.0。

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TC-E 5001

目录号：SY-111069

TC-E 5001 是一种 Wnt 通路抑制剂，通过新型腺苷袋结合抑制端锚聚合酶 1/2 (TNKS1/2)，Kds 值分别为 79 和 28 nM。TC-E 5001 还抑制 Axin2 和 STF，IC50 值分别为 0.709 μM 和 0.215 μM。

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Pep2m, myristoylated

目录号：SY-110116

Cell-permeable, myristoylated form of pep2m. Peptide inhibitor of the interaction between the C-terminus of the GluA2 (AMPA receptor) subunit and N-ethylmaleimide-sensitive fusion protein (NSF), a protein that regulates AMPA receptor function. Reduces pos

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(±)-1,2-Diolein

目录号：SY-110117

(±)-1,2-Diolein (1,2-Dioleoyl-rac-glycerol) 是一种PKC 激活剂，可以增加肌小管 Ca2+内流。

¥1650.00

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6-Deoxyisojacareubin

目录号：SY-110118

6-Deoxyisojacareubin shows moderate inhibitory activity against the QGY-7703 cell line, with the IC50 value of 9.65 uM; it also possesses potency in the inhibition of protein kinase C (PKC).

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Vanicoside A

目录号：SY-110119

Vanicoside A 是一种来自Polygonum pensylvanicum 的蛋白激酶 C (PKC)抑制剂。

¥2618.00

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Kobophenol A

目录号：SY-110120

Kobophenol A has antimicrobial, and anti-inflammatory activities, it might be a candidate for treatment of inflammatory bone diseases relevant to osteoblast cell death. Kobophenol A inhibits AChE activity in a dose-dependent manner, and the IC50 value is

¥1540.00

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SB-747651A Dihydrochloride

目录号：SY-110121

SB-747651A dihydrochloride是一种与ATP竞争性相互作用的抑制剂，特别针对丝裂原和应激激活激酶1 (MSK1)，IC50值为11 nM。此化合物还能抑制PRK2、RSK1、p70S6K和ROCK-II等酶的活性。因其对上述激酶的抑制作用，SB-747651A dihydrochloride在炎症研究中显示出潜力。

¥1694.00

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