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PKCε Inhibitor Scramble Peptide
目录号:SY-110109
PKCε Inhibitor Scramble Peptide为一Scramble肽,其氨基酸序列与PKCε抑制肽相同。
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O-Desmethyl Midostaurin
目录号:SY-110110
O-Desmethyl Midostaurin is the active Midostaurin metabolite via cytochrome P450 liver enzyme metabolism.
¥5698.00
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(-)-Indolactam V
目录号:SY-110111
(-)-Indolactam V is a PKC activator (Kis: 3.36 nM, 1.03 μM for η-CRD2 , γ-CRD2). (-)-Indolactam V also has the Kds are 5.5 nM (η-C1B), 7.7 nM (ε-C1B), 8.3 nM (δ-C1B), 18.9 nM (β-C1A-long), 20.8 nM (α-C1A-long), 137 nM (β-C1B), 138 nM (γ-C1A), 213 nM (γ-C1
¥1386.00
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PKC β pseudosubstrate
目录号:SY-110112
Selective cell-permeable peptide inhibitor of protein kinase C (IC50 ~ 0.5 μM). Consists of amino acids 19 - 31 of PKC pseudosubstrate domain linked by a disulphide bridge to a cell permeabilisation Antennapedia domain vector peptide. The Antennapedia pep
¥2310.00
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Bisindolylmaleimide I HCl
目录号:SY-110113
Bisindolylmaleimide I HCl is a specific ATP-competitive PKC inhibitor.
¥363.00
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PKC-theta inhibitor 1
目录号:SY-110114
PKC-theta inhibitor 1 is an inhibitor of PKCθ (Ki of 6 nM)
¥2442.00
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Dihydrosphingosine
目录号:SY-110115
Dihydrosphingosine is a Protein kinase C inhibitor.
¥1694.00
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Scaff10-8
目录号:SY-108849
Scaff10-8与RhoA结合,抑制了AKAP-Lbc-mediatedRhoA介导的RhoA活化。
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Selisistat
目录号:SY-108850
Selisistat (EX-527) 是一种有效和选择性的 SirT1 (黑腹果蝇中的 Sir2) 抑制剂,IC50 值为 123 nM。Selisistat 缓解多种亨廷顿病动物和细胞模型的病理学。
¥385.00
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