(Rac)-PT2399 is a potent and specific inhibitor of hypoxia-inducible factor 2a (HIF-2α)(IC50 of 0.01 μM).

(S,R,S)-AHPC-C5-COOH (VH032-C5-COOH) is a synthesized E3 ligase ligand-linker conjugate, contains the VH032 VHL-based ligand and a linker to form PROTACs. VH-032 is a selective and potent inhibitor of VHL/HIF-1α interaction with a Kd of 185 nM, has the potential for the study of anemia and ischemic diseases[1].

Diethyl bipy55'DC inhibits CP4H activity in cultured cells. The stability of collagen relies on post-translational modifications, the most prevalent being the hydroxylation of collagen strands by collagen prolyl 4-hydroxylases.

JTZ-951 is a potent and orally active inhibitor of hypoxia inducible factor prolyl hydroxylase (PHD).

Dimethyl-bisphenol A (DMBPA) 是有效的HIF-1α抑制剂，通过从 HIF-1α 解离 Hsp90 促进 HIF-1α 蛋白的降解。Dimethyl-bisphenol A 可降低 Vegfa mRNA 的表达。

Mersalyl is an organic mercurial diuretic.

Atorvastatin lactone 是一种 Atorvastatin 的前药。其中 Atorvastatin 是口服具有活力的 3- 羟基 -3- 甲基戊二酰辅酶 A 还原酶抑制剂。

Simvastatin acid ammonium (Tenivastatin ammonium) 是一种 HMG-CoA 还原酶 (HMGCR) 抑制剂，通过竞争性抑制 HMG-CoA 还原酶（3-羟基-甲基戊二酰辅酶）来减少胆固醇的产生。

(Rac)-5-Keto Fluvastatin (rac 5-Keto Fluvastatin) 是 Fluvastatin 的杂质，Fluvastatin 是一种 HMG-CoA 还原酶的抑制剂。