MK-386 is a potent and selective inhibitor of human type-1 5alpha-reductase.

Isobutyl-deoxynyboquinone (IB-DNQ) is a selective substrate for NAD(P)H: quinone oxidoreductase (NQO1) and is utilized in anticancer research.

Hydroxyevodiamine is a natural product

Danshenol A has strong aldose reductase (AR) inhibitory activity, has IC50 of 0.10 microM which is comparable to that of epalrestat in clinical use. Danshenol A also has antitumor activity in T-24, QGY, K562, Me180 and BIU87 cell lines, shows inhibited growth of K562 (IC50 = 0.53 μg/mL), T-24 (IC50 = 7.94 μg/mL), QGY (IC50 = 4.65 μg/mL) and Me180 (IC50 = 6.89 μg/mL) cell lines.

Tanshindiol B possesses a unique anti-cancer activity whose mechanism involves the inhibition of EZH2 activity and would provide chemically valuable information for designing a new class of potent EZH2 inhibitors. It also possesses the anti-angiogenic act

17alpha-Estradiol-2,4-d2 是 17alpha-Estradiol 的氘代化合物。17alpha-Estradiol 的 CAS 号为 57-91-0。17α-Estradiol 是一种雌性激素，可抑制5α-reductase，在雄原性脱发的研究中有潜力。

8-Lavandulylkaempferol exhibits significant inhibitory effects with IC(50) values of 7.10 and 8.11 microM for butyrylcholinesterase and acetylcholinesterase, respectively. It shows inhibitory activities against aldose reductase, with the the IC50 of 0.79 microM.

Ethyl chlorogenate是一种苯丙素类的天然产物,对大鼠的Aldose Reductase具有抑制活性（IC50=1.5 µM）。

CGP-53153 is a steroidal inhibitor of 5 alpha-reductase (IC50s: 36 and 262 nM in rat and human prostatic tissue).