Imlunestrant (LY-3484356) 是一种口服有效的和选择性的雌激素受体(estrogen receptor)降解剂，能够持续抑制ER依赖基因转录和细胞生长，可用于研究er阳性、her2阴性、esr1突变的晚期或转移性乳腺癌。

Millewanin G shows antiestrogenic activity.

Enclomiphene ((E)-Clomiphene) 是一种有效的、具有口服活性的非甾体雌激素受体 (estrogen receptor) 拮抗剂。Enclomiphene 在睾酮缺乏、男性性腺功能减退症、卵巢功能障碍和 type 2 型糖尿病方面有研究价值。

SNIPER(ER)-87 is a chemical compound composed of a derivative of the inhibitor of apoptosis protein (IAP) ligand LCL161 conjugated to the estrogen receptor α (ERα) ligand 4-hydroxytamoxifen using a PEG linker. It effectively degrades the ERα protein with an IC50 value of 0.097 μM. Within cells, SNIPER(ER)-87 selectively recruits XIAP to ERα, and XIAP functions as the primary E3 ubiquitin ligase responsible for the degradation of ERα induced by SNIPER(ER)-87[1][2].

Clomifene hydrochloride 可以诱导排卵，能够用于不孕症。hydrochloride 是一种简单的、相对安全的、易于给药且耐受性良好的、口服具有活力的化合物。

Psidial A shows activity to enzyme PTP1B; it also reduces tumor growth and stimulate uterus proliferation.

H3B-6545 Hydrochloride is a selective, oral estrogen receptor covalent antagonist (SERCA).

4-Hydroxyestrone 是一种内源性雌激素代谢物，可强烈保护神经元细胞免受氧化损伤。

4-Nonylphenol-d5是4-n-Nonylphenol的氘代标记物，可用于同位素示踪。4-n-Nonylphenol是Nonylphenol ethoxylates(NPEOs)的主要降解物，具有内分泌干扰特性和微弱的雌激素样活性。