AC-261066是一种口服的RARβ2的同型选择性激动剂，pEC50为8.0。

Calcipotriol Impurity C is an impurity of Calcipotriol, a ligand for VDR-like receptors.

VU0155056是一种双重PLD1/2抑制剂, 在体外实验中对PLD1的IC50=81 nM，对PLD2的IC50=240 nM, 在细胞实验中IC50<1 µM，能够抑制乳腺癌细胞侵袭。

Manganese(salen) chloride (EUK-8) 是超氧化物歧化酶和过氧化氢酶的一种模拟物，具有氧自由基清除性能。它可减轻内毒素血症猪的急性肺损伤。

(24S)-24,25-Dihydroxyvitamin D3 undergoes multiple hydroxylation processes to form active vitamin D3 analogs.

ROC-0929 (compound 13a) is a potent and selective inhibitor of secreted phospholipases A2 (sPLA2s), effectively targeting hGX with an IC50 of 80 nM. It efficiently inhibits the phosphorylation of ERK1/2 and p-38. sPLA2s, belonging to the disulfide-rich, Ca2+-dependent enzyme family, catalyze the hydrolysis of glycero-phospholipids at the sn-2 position, resulting in the release of a fatty acid and a lysophospholipid. ROC-0929 holds promise in researching inflammation-related diseases.

Luciferase 是一种在生物发光细菌中发现的依赖黄素的单加氧酶。 Luciferase 是识别和表征功能变体的宝贵工具，可用于研究基因表达、细胞内信号传导、转录因子、受体活性和蛋白质折叠。

SR1555 is a selective RORγ inverse agonist that inhibits the development and function of TH17 cells, a subset of T cells that have been involved in the pathology of several autoimmune diseases such as rheumatoid arthritis and multiple sclerosis.

V-125 is an agonist of retinoid X receptors.