PKM2 inhibitor G是丙酮酸激酶抑制剂。

L-6355 is an agent of bioactive chemicals.

4-Nitrophenyl phenylphosphonate is a substrate for 5'-nucleotide phosphodiesterases. It is a more preferable substrate to 5'-nucleotide phosphodiesterases than naturally occurring nucleotides or bis(4-nitrophenyl) phosphate because of its stability, ease of synthesis, and higher rate of hydrolysis under saturating conditions.

Alkannin 是一种有效且特异性的肿瘤型丙酮酸激酶-M2 (PKM2) 抑制剂，不抑制 PKM1 和丙酮酸激酶-L (PKL)。Alkannin 是一种潜在的抗癌剂。

ITI-214 free base is a picomolar PDE1 inhibitor with excellent selectivity against other PDE family members and against a panel of enzymes, receptors, transporters, and ion channels, exhibits potent PDE1 inhibitory activity (Ki = 58 pM).

Enpp-1-IN-5 是一种有效的外核苷酸焦磷酸酶-磷酸二酯酶 1 (enpp-1) 抑制剂。ENPP 1 显示出广泛的特异性，能够切割多种底物（包括核苷酸和核苷酸糖的磷酸二酯键、核苷酸和核苷酸糖的焦磷酸键）。 Enpp-1-IN-5 具有潜力进行癌症和传染病的研究。

PKM2-IN-3 is a potent PKM2 kinase inhibitor, displaying an IC 50 value of 4.1 μM. The compound effectively suppresses PKM2-mediated glycolysis and NLRP3 activation, thereby exerting an anti-neuroinflammatory effect.

PKM2 activator 2是一种丙酮酸激酶 M2（PKM2）激活剂，AC 50 值为 66 nM。PKM2 activator 2具有抗肿瘤增殖和缓解沃伯格效应的作用，通过激活 PKM2 使细胞的糖酵解代谢恢复正常。

11-Oxoisomogroside V 是从罗汉果(Siraitia grosvenorii)中分离得到的三萜类糖苷化合物，具有抗氧化和抗炎活性。11-Oxoisomogroside V 可激活 PGC-1α 的转录活性。11-Oxoisomogroside V 可提高荧光素酶活性。