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Acetylene-linker-Val-Cit-PABC-MMAE
目录号:SY-101362
Acetylene-linker-Val-Cit-PABC-MMAE (LCB14-0602) is a drug-linker conjugate for antibody-drug conjugates (ADCs) that combines the ADC linker (Acetylene-linker-Val-Cit-PABC) with the potent tubulin inhibitor MMAE.
¥1725.00
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Mal-(CH2)5-Val-Cit-PAB-Eribulin
目录号:SY-101361
Mal-(CH2)5-Val-Cit-PAB-Eribulin is a potent antitumor ADC drug-linker conjugate that utilizes Eribulin, an anti-microtubule agent, connected through the Mal-(CH2)5-Val-Cit-PAB linker.
¥5118.00
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MC-Val-Cit-PAB-carfilzomib iodide
目录号:SY-101360
MC-Val-Cit-PAB-carfilzomib is a potent antitumor drug-linker conjugate for antibody-drug conjugates (ADC), comprising the irreversible proteasome inhibitor carfilzomib, connected through the ADC linker MC-Val-Cit-PAB.
¥3910.00
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PAC
目录号:SY-101367
PAC is a chemical conjugate consisting of an ADCs linker and PROTACs linked to an antibody. When PAC is conjugated to an antibody, it exhibits enhanced degradation of estrogen receptor-alpha (ERα) in comparison to PROTAC alone.
¥5852.00
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MC-Gly-Gly-Phe-Gly-(S)-Cyclopropane-Exatecan
目录号:SY-101366
MC-Gly-Gly-Phe-Gly-(R)-Cyclopropane-Exatecan 是抗体偶联活性分子的一部分 (drug-linker conjugate for ADC),包含 Exatecan 。Exatecan 是一种 DNA 拓扑异构酶 I (Topoisomerase I) 抑制剂 (IC50=2.2 μM)。
¥8625.00
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MC-(β-Ala)-PABC-(β-D-GlcUA)-amide-PEG1-CH2-CC-885
目录号:SY-101368
Comp Ie (MC-(β-Ala)-PABC-(β-D-GlcUA)-amide-PEG1-CH2-CC-885) 为一种新型抗体新降解剂偶联活性分子 (AnDC) 的合成降解剂偶联物。
¥10350.00
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