hMCH-1R antagonist 1

目录号：SY-112267

hMCH-1R antagonist 1 (Compound 30)为高效且具有选择性的hMCHR1拮抗剂，KB值仅为3.6 nM。它与hMCHR1和hMCHR2的结合能力强，IC50值分别为65 nM与49 nM，主要用于代谢研究领域。

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GPR35 agonist 5

目录号：SY-112268

GPR35 agonist5（3,5-dinitro-bisphenol A; compound 6）作为一种弱GPR35激动剂，能够将CHO-S细胞阻滞在G1/Go期。

¥2012.00

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ATC0065 HCl

目录号：SY-112269

ATC0065 dihydrochloride is a novel nonpeptidic and potent melanin-concentrating hormone receptor 1 (MCHR1) selective antagonist.

¥1610.00

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BigLEN(mouse)

目录号：SY-112270

GPR171 agonist. ProSAAS-derived neuropeptide. Regulates food intake in mice. Inhibits the release of glutamate onto parvocellular neurons of the paraventricular nucleus in a process dependent upon activation of postsynaptic G proteins.

¥516.00

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GPR40 Activator 2

目录号：SY-112271

GPR40 Activator 2 is a highly effective activator of the GPR40 receptor.

¥1127.00

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GPR40 agonist 6

目录号：SY-112272

GPR40 agonist 6 (Compound 7a) 是游离脂肪酸受体 1的选择性激动剂（FFAR1或GPR40），其对于GPR40的EC50值为 0.058 μM。

¥621.00

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Melanin Concentrating Hormone, salmon

目录号：SY-112273

Melanin Concentrating Hormone (MCH), a 19 amino acid cyclic peptide, is largely expressed in the hypothalamus.

¥2288.00

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GPR40 Activator 1

目录号：SY-112274

GPR40 Activator 1 is a potent GPR40 activator for treatment of type 2 diabetes.

¥3266.00

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GPR119 agonist 2

目录号：SY-112275

GPR119 agonist2（化合物43）是一种口服活性的GPR119激动剂。在啮齿动物中表现出优良的药代动力学特性，并能有效提高小鼠和大鼠的葡萄糖耐受性。GPR119 agonist2有望用于研究II型糖尿病。

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