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GPR4 antagonist 1
目录号:SY-112249
GPR4 antagonist 1 is a GPR4 antagonist (IC50: 189 nM).
¥2668.00
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BMS-819881
目录号:SY-112250
BMS-819881 is a melaninconcentrating hormone receptor 1 (MCHR1) antagonist, which binds rat MCHR1 with a Ki of 7 nM and it also is selective and potent for CYP3A4 activity with an EC50 of 13 μM.
¥3749.00
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Kisspeptin-14 human
目录号:SY-112251
Kisspeptin-14 human是Kisspeptin的活性片段短肽,含有14个氨基酸,由KiSS-1基因编码。Kisspeptin-14 human是一种GPR54激动剂,在CHO-K1细胞上对人和大鼠GPR54受体的Ki值分别为1.65和2.04 nM,EC50值分别为7.22和1.33 nM。
¥575.00
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CATPB
目录号:SY-112252
CATPB is a novel inverse hFFA2 agonist.
¥471.00
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Pyrone-211
目录号:SY-112253
Pyrone-211 是一种有效的 GPR84 激动剂和 AKR1C3 抑制剂,参与扩展的多胺途径。
¥2208.00
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DHICA
目录号:SY-112254
DHICA (5,6-Dihydroxyindole-2-carboxylic acid) 作为黑色素合成的中间体及真黑色素的关键成分,此外它还能作为GPR35的中等效力激动剂。在 U2OS 细胞系中,DHICA能以 23.2 μM 的EC50值促进β-arrestin的转位信号。此化合物对于促进和保护 DNA 损伤具有显著作用。
¥297.00
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BMS-986034
目录号:SY-112255
BMS-986034 is a GPR119 agonist.
询价
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NGD-4715
目录号:SY-112256
NGD-4715 is a selective and orally active antagonist of melanin-concentrating hormone receptor 1.
询价
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(S)-CVN424
目录号:SY-112257
(S)-CVN424 is a powerful modulator of G-Protein-Coupled Receptor 6 (GPR6), known for its involvement in neurological and psychiatric disorders research, such as Parkinson's disease.
¥5175.00
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