Cyprodinil 是一种苯胺嘧啶广谱杀菌剂，可抑制植物病原真菌蛋氨酸的生物合成。Cyprodinil 抑制B. cinerea，P. herpotrichoides，H. oryzae 的菌丝体细胞在无氨基酸的培养基上生长，IC50s 分别为 0.44，4.8，0.03 μM。在没有 AR 激动剂 DHT 的情况下，Cyprodinil 充当雄激素受体 (AR) 激动剂 (EC50=1.91 μM)，并抑制 DHT 的雄激素作用 (IC50=15.1 μM)。

non-steroidal androgen receptor (AR) antagonist

11-Ketodihydrotestosterone is a metabolite of 11β-Hydroxyandrostenedione. It is an active androgen and is also a potent androgen receptor (AR) agonist (Ki: 20.4 nM, EC50: 1.35 nM for human AR).

(R)-Bicalutamide 是一种 Bicalutamide 的 R 型对映体，是一种雄激素受体 (AR) 拮抗剂，表现出抗肿瘤效果。(R)-Bicalutamide 广泛的用于前列腺癌的研究。

Leelamine hydrochloride, a tricyclic diterpene extracted from pine tree bark, inhibits the transcriptional activity of the androgen receptor, known to regulate fatty acid synthesis [2,3]. This compound acts as a cannabinoid receptor type 1 (CB1) agonist and suppresses SREBP1-regulated fatty acid/lipid synthesis in prostate cancer cells, irrespective of androgen receptor status.

Dehydroepiandrosterone-d2 是 Dehydroepiandrosterone 的氘代化合物。