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Neuropeptide EI, rat
目录号:SY-112240
Displays functional MCH-antagonist and MSH-agonist activity in different behavioral paradigms.
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[Ala17]-MCH
目录号:SY-112241
Potent melanin-concentrating hormone (MCH) receptor agonist (EC50 values are 17 and 54 nM at MCH1 and MCH2 receptors respectively). Displays some selectivity towards MCH1 over MCH2 (Ki values are 0.16 and 34 nM respectively).
¥2530.00
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AMG 837 hemicalcium
目录号:SY-112242
AMG 837 hemicalcium 是一种有效的、口服具有活力的 GPR40/FFA1部分激动剂。AMG 837 hemicalcium 能够抑制 [3H]AMG 837 与人类 FFA1受体的特异性结合 (pIC50: 8.13)。AMG 837 hemicalcium 能够提高啮齿动物的胰岛素分泌,减少葡萄糖水平。
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[Orn8]-Urotensin II
目录号:SY-112243
[Orn8]-Urotensin II 是一种 Urotensin 受体配体和 Urotensin 受体的部分激动剂。
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RTI-13951-33
目录号:SY-112244
RTI-13951-33 is an effective and brain-penetrant GPR88 agonist (EC50: 25 nM, in GPR88 cAMP functional assay).
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BigLEN(rat)
目录号:SY-112245
Potent GPR171 agonist (EC50 = 1.6 nM). ProSAAS-derived peptide. Regulates body weight in mice and promotes the outgrowth of neurites in Neuro2A cells.
¥2185.00
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AM-5262
目录号:SY-112246
AM-5262 is a potent GPR40 Full Agonist with improved rat PK profile and general selectivity profile.
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AMG7703
目录号:SY-112247
AMG7703 is a bioactive chemical.
¥1863.00
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MCH-1 antagonist 1
目录号:SY-112248
MCH-1 antagonist 1 also inhibits CYP3A4 (IC50: 10μM).MCH-1 antagonist 1 is a potent melanin concentrating hormone (MCH-1) antagonist (Ki: 2.6 nM).
¥5256.00
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